Cavalluzzi, Maria M.: search on Z-Library

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1

Ligand efficiency metrics in drug discovery: the pros and cons from a practical perspective

Cavalluzzi, Maria Maddalena, Mangiatordi, Giuseppe Felice, Nicolotti, Orazio, Lentini, Giovanni

Journal:

Expert Opinion on Drug Discovery

Year:

2017

Language:

english

File:

PDF, 1.79 MB

english, 2017

2

Insights on Molecular Determinants of hERG K+ Channel Inhibition: Design, Synthesis, and Biological Evaluation of Lubeluzole Derivatives

Gualdani, Roberta, Cavalluzzi, Maria Maddalena, Tadini-Buoninsegni, Francesco, Moncelli, Maria Rosa, Lentini, Giovanni

Journal:

Biophysical Journal

Year:

2015

Language:

english

File:

PDF, 46 KB

english, 2015

3

Facile, alternative route to Lubeluzole, its enantiomer, and the racemate

Claudio Bruno, Alessia Carocci, Alessia Catalano, Maria M. Cavalluzzi, Filomena Corbo, Carlo Franchini, Giovanni Lentini, Vincenzo Tortorella

Journal:

Year:

2006

Language:

english

File:

PDF, 110 KB

english, 2006

4

Microwave-Assisted Synthesis of KN-93, a Potent and Selective Inhibitor of Ca²+/Calmoduline-Dependent Protein Kinase II

Bruno, Claudio, Lentini, Giovanni, Catalano, Alessia, Carocci, Alessia, Lovece, Angelo, Di Mola, Antonia, Cavalluzzi, Maria, Tortorella, Paolo, Loiodice, Fulvio, Iaccarino, Guido, Campiglia, Pietro, N

Journal:

Year:

2010

Language:

english

File:

PDF, 128 KB

english, 2010

5

Discovery of a new mexiletine-derived agonist of the hERG K + channel

Gualdani, Roberta, Cavalluzzi, Maria Maddalena, Tadini-Buoninsegni, Francesco, Lentini, Giovanni

Journal:

Biophysical Chemistry

Year:

2017

Language:

english

File:

PDF, 623 KB

english, 2017

6

Synthesis and evaluation of berberine derivatives and analogs as potential antiacetylcholinesterase and antioxidant agents

Roselli, Mariagrazia, Cavalluzzi, Maria Maddalena, Bruno, Claudio, Lovece, Angelo, Carocci, Alessia, Franchini, Carlo, Habtemariam, Solomon, Lentini, Giovanni

Journal:

Phytochemistry Letters

Year:

2016

Language:

english

File:

PDF, 778 KB

english, 2016

7

First synthesis and full characterization of mexiletine N-carbonyloxy β-d-glucuronide

Maria Maddalena Cavalluzzi, Giovanni Lentini, Angelo Lovece, Claudio Bruno, Alessia Catalano, Alessia Carocci, Carlo Franchini

Journal:

Tetrahedron Letters

Year:

2010

Language:

english

File:

PDF, 332 KB

english, 2010

8

Combined Modifications of Mexiletine Pharmacophores for New Lead Blockers of Nav1.4 Channels

De Bellis, Michela, De Luca, Annamaria, Desaphy, Jean F., Carbonara, Roberta, Heiny, Judith A., Kennedy, Ann, Carocci, Alessia, Cavalluzzi, Maria M., Lentini, Giovanni, Franchini, Carlo, Conte Camerin

Journal:

Biophysical Journal

Year:

2013

Language:

english

File:

PDF, 564 KB

english, 2013

9

Nitro-substituted tetrahydroindolizines and homologs: Design, kinetics, and mechanism of α-glucosidase inhibition

Tavani, Cinzia, Bianchi, Lara, De Palma, Annalisa, Passeri, Giovanna Ilaria, Punzi, Giuseppe, Pierri, Ciro Leonardo, Lovece, Angelo, Cavalluzzi, Maria Maddalena, Franchini, Carlo, Lentini, Giovanni, P

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2017

Language:

english

File:

PDF, 2.00 MB

english, 2017

10

Ultrasound and deep eutectic solvents: An efficient combination to tune the mechanism of steviol glycosides extraction

Milani, Gualtiero, Vian, Maryline, Cavalluzzi, Maria Maddalena, Franchini, Carlo, Corbo, Filomena, Lentini, Giovanni, Chemat, Farid

Journal:

Ultrasonics Sonochemistry

Year:

2020

File:

PDF, 2.25 MB

2020

11

The Chemistry and Pharmacology of Citrus Limonoids

Gualdani, Roberta, Cavalluzzi, Maria, Lentini, Giovanni, Habtemariam, Solomon

Journal:

Year:

2016

Language:

english

File:

PDF, 4.45 MB

english, 2016

12

Human ether-à-go-go-related potassium channel: exploring SAR to improve drug design

Cavalluzzi, Maria Maddalena, Imbrici, Paola, Gualdani, Roberta, Stefanachi, Angela, Mangiatordi, Giuseppe Felice, Lentini, Giovanni, Nicolotti, Orazio

Journal:

Drug Discovery Today

Year:

2019

Language:

english

File:

PDF, 4.30 MB

english, 2019

13

A Focus on the Synthesis and Pharmacokinetics of Tocainide and its Analogues

Carocci, Alessia, Corbo, Filomena, Lentini, Giovanni, Cavalluzzi, Maria Maddalena, Franchini, Carlo, Catalano, Alessia

Journal:

Current Medicinal Chemistry

Year:

2019

File:

PDF, 733 KB

2019

14

A convenient synthesis of lubeluzole and its enantiomer: Evaluation as chemosensitizing agents on human ovarian adenocarcinoma and lung carcinoma cells

Cavalluzzi, Maria Maddalena, Viale, Maurizio, Bruno, Claudio, Carocci, Alessia, Catalano, Alessia, Carrieri, Antonio, Franchini, Carlo, Lentini, Giovanni

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2013

Language:

english

File:

PDF, 618 KB

english, 2013

15

The chemosensitizing agent lubeluzole binds calmodulin and inhibits Ca2+/calmodulin-dependent kinase II

Bruno, Claudio, Cavalluzzi, Maria Maddalena, Rusciano, Maria Rosaria, Lovece, Angelo, Carrieri, Antonio, Pracella, Riccardo, Giannuzzi, Giulia, Polimeno, Lorenzo, Viale, Maurizio, Illario, Maddalena,

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 1.03 MB

english, 2016

16

Lubeluzole: from anti-ischemic drug to preclinical antidiarrheal studies

Cavalluzzi, Maria Maddalena, Budriesi, Roberta, De Salvia, Maria Antonietta, Quintieri, Laura, Piarulli, Monica, Milani, Gualtiero, Gualdani, Roberta, Micucci, Matteo, Corazza, Ivan, Rosato, Antonio,

Journal:

Pharmacological Reports

Year:

2020

File:

PDF, 1.30 MB

2020

17

Hydroxylated Analogs of Mexiletine as Tools for Structural-Requirements Investigation of the Sodium Channel Blocking Activity

Alessia Catalano, Alessia Carocci, Maria M. Cavalluzzi, Antonia Di Mola, Giovanni Lentini, Angelo Lovece, Antonella Dipalma, Teresa Costanza, Jean-François Desaphy, Diana Conte Camerino, Carlo Franchi

Journal:

Archiv der Pharmazie

Year:

2010

Language:

english

File:

PDF, 486 KB

english, 2010

18

Searching for new antiarrhythmic agents: Evaluation of meta-hydroxymexiletine enantiomers

Catalano, Alessia, Budriesi, Roberta, Bruno, Claudio, Di Mola, Antonia, Defrenza, Ivana, Cavalluzzi, Maria Maddalena, Micucci, Matteo, Carocci, Alessia, Franchini, Carlo, Lentini, Giovanni

Journal:

European Journal of Medicinal Chemistry

Year:

2013

Language:

english

File:

PDF, 299 KB

english, 2013

19

2-Arylazetidines as ligands for nicotinic acetylcholine receptors

Degennaro, Leonardo, Zenzola, Marina, Laurino, Annunziatina, Cavalluzzi, Maria Maddalena, Franchini, Carlo, Habtemariam, Solomon, Matucci, Rosanna, Luisi, Renzo, Lentini, Giovanni

Journal:

Chemistry of Heterocyclic Compounds

Year:

2017

Language:

english

File:

PDF, 268 KB

english, 2017

20

An Improved Synthesis of m-Hydroxymexiletine, a Potent Mexiletine Metabolite

Catalano, Alessia, Carocci, Alessia, Lentini, Giovanni, Defrenza, Ivana, Maddalena Cavalluzzi, Maria, Franchini, Carlo

Journal:

Drug Metabolism Letters

Year:

2012

Language:

english

File:

PDF, 334 KB

english, 2012

21

Synthesis, antiarrhythmic activity, and toxicological evaluation of mexiletine analogues

Roselli, Mariagrazia, Carocci, Alessia, Budriesi, Roberta, Micucci, Matteo, Toma, Maddalena, Di Cesare Mannelli, Lorenzo, Lovece, Angelo, Catalano, Alessia, Cavalluzzi, Maria Maddalena, Bruno, Claudio

Journal:

European Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 493 KB

english, 2016

22

Antioxidant Activity of Uva di Troia Canosina: Comparison of Two Extraction Methods

Roselli, Mariagrazia, Lovece, Angelo, Bruno, Claudio, Maddalena Cavalluzzi, Maria, Laghezza, Antonio, Mercurio, Annalisa, Lentini, Giovanni, Corbo, Filomena, la Forgia, Flavia, Fontana, Sergio, Habtem

Journal:

Clinical Immunology Endocrine & Metabolic Drugs

Year:

2015

Language:

english

File:

PDF, 462 KB

english, 2015

23

Lactoferrin-Derived Peptides as a Control Strategy against Skinborne Staphylococcal Biofilms

Quintieri, Laura, Caputo, Leonardo, Monaci, Linda, Cavalluzzi, Maria Maddalena, Denora, Nunzio

Journal:

Year:

2020

File:

PDF, 1.86 MB

2020

24

Synthesis and evaluation of voltageâgated sodium channel blocking pyrroline derivatives endowed with both antiarrhythmicÂ and antioxidant activities

Carocci, Alessia, Budriesi, Roberta, Micucci, Matteo, Cavalluzzi, Maria Maddalena, Milani, Gualtiero, Catalano, Alessia, De Palma, Annalisa, Corbo, Filomena, Franchini, Carlo, Habtemariam, Solomon, Gi

Journal:

Year:

2020

File:

PDF, 1.24 MB

2020

25

Chiral Aryloxyalkylamines: Selective 5-HT1B/1D Activation and Analgesic Activity

Alessia Carocci, Giovanni Lentini, Alessia Catalano, Maria Maddalena Cavalluzzi, Claudio Bruno, Marilena Muraglia, Nicola Antonio Colabufo, Nicoletta Galeotti, Filomena Corbo, Rosanna Matucci, Carla G

Journal:

Year:

2010

Language:

english

File:

PDF, 350 KB

english, 2010

26

Antimicrobial and Antibiofilm Activities of Citrus Water-Extracts Obtained by Microwave-Assisted and Conventional Methods

Caputo, Leonardo, Quintieri, Laura, Cavalluzzi, Maria, Lentini, Giovanni, Habtemariam, Solomon

Journal:

Year:

2018

Language:

english

File:

PDF, 1.81 MB

english, 2018

27

Molecular Determinants of Human Voltage-Gated Sodium Channels Blockade by Lubeluzole

Desaphy, Jean-François, Costanza, Teresa, Carbonara, Roberta, Maddalena Cavalluzzi, Maria, Franchini, Carlo, Lentini, Giovanni, Conte Camerino, Diana

Journal:

Biophysical Journal

Year:

2012

Language:

english

File:

PDF, 41 KB

english, 2012

28

Molecular Insights into hERG Potassium Channel Blockade by Lubeluzole

Gualdani, Roberta, Cavalluzzi, Maria Maddalena, Tadini-Buoninsegni, Francesco, Convertino, Marino, Gailly, Philippe, Stary-Weinzinger, Anna, Lentini, Giovanni

Journal:

Cellular Physiology and Biochemistry

Year:

2018

Language:

english

File:

PDF, 1.98 MB

english, 2018

29

New N-(phenoxydecyl)phthalimide derivatives displaying potent inhibition activity towards α-glucosidase

Rossana Pascale, Alessia Carocci, Alessia Catalano, Giovanni Lentini, Anna Spagnoletta, Maria Maddalena Cavalluzzi, Francesco De Santis, Annalisa De Palma, Vito Scalera, Carlo Franchini

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 551 KB

english, 2010

30

Preparation of (−)-(R)-2-(2,3,4,5,6-pentafluorophenoxy)-2-(phenyl-d5)acetic acid: an efficient 1H NMR chiral solvating agent for direct enantiomeric purity evaluation of quinoline-containing antimalarial drugs

Cavalluzzi, Maria Maddalena, Lovece, Angelo, Bruno, Claudio, Franchini, Carlo, Lentini, Giovanni

Journal:

Tetrahedron: Asymmetry

Year:

2014

Language:

english

File:

PDF, 1.11 MB

english, 2014

31

One-step synthesis of homochiral O-aryl and O-heteroaryl mandelic acids and their use as efficient 1H NMR chiral solvating agents

Maria Maddalena Cavalluzzi, Claudio Bruno, Giovanni Lentini, Angelo Lovece, Alessia Catalano, Alessia Carocci, Carlo Franchini

Journal:

Tetrahedron: Asymmetry

Year:

2009

Language:

english

File:

PDF, 796 KB

english, 2009

32

Synthesis of (R)-, (S)-, and (RS)-hydroxymethylmexiletine, one of the major metabolites of mexiletine

Maria Maddalena Cavalluzzi, Alessia Catalano, Claudio Bruno, Angelo Lovece, Alessia Carocci, Filomena Corbo, Carlo Franchini, Giovanni Lentini, Vincenzo Tortorella

Journal:

Tetrahedron: Asymmetry

Year:

2007

Language:

english

File:

PDF, 198 KB

english, 2007

33

Optically Active Mexiletine Analogues as Stereoselective Blockers of Voltage-Gated Na + Channels

Franchini, Carlo, Carocci, Alessia, Catalano, Alessia, Cavalluzzi, Maria M., Corbo, Filomena, Lentini, Giovanni, Scilimati, Antonio, Tortorella, Paolo, Camerino, Diana Conte, Luca, Annamaria De

Journal:

Journal of Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 162 KB

english, 2003

34

Stereoselective Modulation of P-Glycoprotein by Chiral Small Molecules

Carocci, Alessia, Catalano, Alessia, Turi, Francesco, Lovece, Angelo, Cavalluzzi, Maria M., Bruno, Claudio, Colabufo, Nicola A., Contino, Marialessandra, Perrone, Maria G., Franchini, Carlo, Lentini,

Journal:

Year:

2016

Language:

english

File:

PDF, 522 KB

english, 2016

35

The Crystal Structure of N-[(2E)-3-(4-Chlorophenyl)prop-2-en-1-yl]-4-methoxy-N-methylbenzenesulfonamide

Carrozzini, Benedetta, Belviso, Benny Danilo, Bruno, Claudio, Cavalluzzi, Maria Maddalena, Lovece, Angelo, Lentini, Giovanni, Caliandro, Rocco

Journal:

Journal of Chemical Crystallography

Year:

2018

Language:

english

File:

PDF, 1.47 MB

english, 2018

36

(S)-Ethyl 2-(tert-butoxycarbonylamino)-3-(2-iodo-4,5-methylenedioxyphenyl)propanoate

Lentini, Giovanni, Cavalluzzi, Maria, Degennaro, Leonardo, Fracchiolla, Giuseppe, Perna, Filippo, Scilimati, Antonio

Journal:

Year:

2019

File:

PDF, 764 KB

2019

37

COVID-19, Chloroquine Repurposing, and Cardiac Safety Concern: Chirality Might Help

Lentini, Giovanni, Cavalluzzi, Maria Maddalena, Habtemariam, Solomon

Journal:

Year:

2020

File:

PDF, 361 KB

2020

38

N-(Phenoxyalkyl)amides as MT1 and MT2 ligands: Antioxidant properties and inhibition of Ca2+/CaM-dependent kinase II

Carocci, Alessia, Catalano, Alessia, Bruno, Claudio, Lovece, Angelo, Roselli, Maria Grazia, Cavalluzzi, Maria Maddalena, De Santis, Francesco, De Palma, Annalisa, Rusciano, Maria Rosaria, Illario, Mad

Journal:

Bioorganic & Medicinal Chemistry

Year:

2013

Language:

english

File:

PDF, 235 KB

english, 2013

39

Optically Active Mexiletine Analogues as Stereoselective Blockers of Voltage-Gated Na + Channels.

Franchini, Carlo, Carocci, Alessia, Catalano, Alessia, Cavalluzzi, Maria M., Corbo, Filomena, Lentini, Giovanni, Scilimati, Antonio, Tortorella, Paolo, Camerino, Diana Conte, De Luca, Annamaria

Journal:

Journal of Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 41 KB

english, 2005

40

Pilsicainide and Its Oxymethylene Analog: Facile Alternative Syntheses and in vitro Testing on Human Skeletal Muscle Sodium Channels

Lentini, Giovanni, Bruno, Claudio, Catalano, Alessia, Desaphy, Jean-Francois, M. Cavalluzzi, Maria, Carocci, Alessia, Dipalma, Antonella, Franchini, Carlo, Conte Camerino, Diana, Tortorella, Vincenzo

Journal:

Year:

2007

Language:

english

File:

PDF, 194 KB

english, 2007

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